Interaction between iodothyronines and thyrotropin receptor in human cultured thyroid cells

J Recept Res. 1981;2(4):367-82. doi: 10.3109/107998981809038873.

Abstract

In order to verify the existence of a "short-loop" negative feedback between iodothyronines and adenylate cyclase system of human thyroid, we have studied the effect of preincubation with iodothyronines, iodotyrosines, iodothyronine analogues and iodide on TSH-induced cAMP cellular accumulation in normal human thyroid cells in primary culture. Iodide did not produce an inhibitory effect on TSH-dependent adenylate cyclase system both in normal human thyroid plasma membranes and cultured cells. Iodothyronines at a 30-40 microM concentration did not inhibit the TSH-dependent adenylate cyclase activity of human thyroid plasma membranes; however at a 1 microM concentration they were able to inhibit the TSH-dependent cAMP accumulation by cultured cells. Preincubation with iodotyrosines and iodothyronine analogues failed to inhibit the TSH-responsive cAMP accumulation in human thyroid cultured cells.

Publication types

  • Comparative Study

MeSH terms

  • Adenylyl Cyclases / metabolism
  • Adrenal Cortex / metabolism
  • Adrenocorticotropic Hormone / pharmacology
  • Cells, Cultured
  • Dinoprostone
  • Humans
  • Iodides / pharmacology
  • Prostaglandins E / pharmacology
  • Receptors, Cell Surface / drug effects*
  • Receptors, Thyrotropin
  • Thyroid Gland / metabolism*
  • Thyroid Hormones / pharmacology*
  • Thyrotropin / pharmacology

Substances

  • Iodides
  • Prostaglandins E
  • Receptors, Cell Surface
  • Receptors, Thyrotropin
  • Thyroid Hormones
  • Adrenocorticotropic Hormone
  • Thyrotropin
  • Adenylyl Cyclases
  • Dinoprostone