Panax ginseng and Eleuthrococcus senticosus extracts--in vitro studies on binding to steroid receptors

Endocrinol Jpn. 1982 Oct;29(5):567-73. doi: 10.1507/endocrj1954.29.567.

Abstract

We have examined the binding of 44% saponin from Panax ginseng, and extracts from Eluthrococcus senticosus (Siberian ginseng) to classical steroid receptors in vitro. Both extracts had demonstrable affinity for progestin, mineralocorticoid and glucocorticoid receptors; the Siberian ginseng also bound to estrogen receptors. Highest affinity binding was to glucocorticoid receptors, with an approximate Ki of 8 x 10(-6) M for Panax ginseng. Such interactions may explain the reported glucocorticoid-like effects of ginseng in vivo.

MeSH terms

  • Animals
  • Binding, Competitive / drug effects
  • Female
  • In Vitro Techniques
  • Kidney / metabolism
  • Mice
  • Panax* / metabolism
  • Plants, Medicinal*
  • Rats
  • Rats, Inbred Strains
  • Receptors, Estrogen / metabolism
  • Receptors, Glucocorticoid / metabolism
  • Receptors, Mineralocorticoid
  • Receptors, Steroid / metabolism*
  • Saponins / metabolism
  • Uterus / metabolism

Substances

  • Receptors, Estrogen
  • Receptors, Glucocorticoid
  • Receptors, Mineralocorticoid
  • Receptors, Steroid
  • Saponins