Synthesis of benzo-benzothiopyranoquinolines (pyridobenzothioxanthones) as possible schistosomicidal and antitumor agents

Pharmazie. 1978 Jul;33(7):424-6. doi: 10.1002/chin.197849249.

Abstract

The synthesis of a new class of compounds structurally related to cyclohexenothiaxanthones and benzothiaxanthones including a pyridine ring is described in an attempt to find compounds that may have schistosomicidal and carcinostatic activity. Synthesis was achieved through the condensation of amino-cyclohexenothiaxanthones and amino-benzothiaxanthones with ethyl acetoacetate by the Knorr and Conrad-Limpach methods.

MeSH terms

  • Animals
  • Antineoplastic Agents
  • Chemical Phenomena
  • Chemistry
  • Methods
  • Quinolines / chemical synthesis*
  • Quinolines / pharmacology
  • Schistosomicides

Substances

  • Antineoplastic Agents
  • Quinolines
  • Schistosomicides