Comparative carcinogenicity in F344 rats of the tobacco-specific nitrosamines, N'-nitrosonornicotine and 4-(N-methyl-N-nitrosamino)-1-(3-pyridyl)-1-butanone

Cancer Res. 1980 Feb;40(2):298-302.

Abstract

The tobacco-specific carcinogens, N'-nitrosonornicotine (NNN) and 4-(N-methyl-N-nitrosamino)-1-(3-pyridyl)-1-butanone (NNK), were tested for carcinogenicity in F344 rats. Each nitrosamine in trioctanoin was administered by s.c. injection to 12 male and 12 female rats over a period of 20 weeks. The total dose of each nitrosamine was 3.4 mmol. The experiment was terminated after 12 months. NNK induced nasal cavity tumors in 83% of the males and in 83% of the females, liver tumors in 83% of the males and in 100% of the females, and lung tumors in 67% of the males and in 67% of the females. NNN induced nasal cavity tumors in 92% of the males and in 75% of the females. Only one liver tumor and no lung tumors were observed in the NNN-treated rats. These results indicate that, in the F344 rat, NNK is a more powerful carcinogen than is NNN.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Carcinogens*
  • Female
  • Liver Neoplasms / chemically induced
  • Lung Neoplasms / chemically induced
  • Male
  • Nasal Cavity
  • Neoplasms, Experimental / chemically induced*
  • Neoplasms, Experimental / pathology
  • Nicotiana*
  • Nicotine / analogs & derivatives*
  • Nicotine / toxicity
  • Nitrosamines / toxicity*
  • Nose Neoplasms / chemically induced
  • Plants, Toxic*
  • Pyridines / toxicity
  • Rats
  • Rats, Inbred F344

Substances

  • Carcinogens
  • Nitrosamines
  • Pyridines
  • Nicotine
  • 4-(N-methyl-N-nitrosamino)-1-(3-pyridyl)-1-butanone
  • N'-nitrosonornicotine