Antiallergy activity of 10-oxo-10-H-pyridazino[6,1-b]quinazoline-2-carboxylic acids

J Med Chem. 1980 Aug;23(8):964-6. doi: 10.1021/jm00182a030.

Abstract

A series of substituted 10-oxo-10H-pyridazino[6,1-b]quinazoline-2-carboxylic acids was prepared and evaluated as antiallergy agents. The 8-chloro and unsubstituted analogues were more potent that cromolyn sodium and doxantrazole intravenously in the rat PCA test. None of the analogues possessed significant oral activity.

MeSH terms

  • Animals
  • Hypersensitivity / drug therapy*
  • Passive Cutaneous Anaphylaxis / drug effects
  • Pyridazines / chemical synthesis
  • Pyridazines / pharmacology
  • Quinazolines / chemical synthesis*
  • Quinazolines / pharmacology
  • Rats
  • Structure-Activity Relationship

Substances

  • Pyridazines
  • Quinazolines