Calpain inhibitors reduce depolarization induced loss of tau protein in primary septo-hippocampal cultures

Neurosci Lett. 1995 Jul 21;194(3):149-52. doi: 10.1016/0304-3940(95)11745-i.

Abstract

We studied the effects of a 6-min potassium depolarization injury produced by 60 mM KCl and 1.8 mM or 5.8 mM extracellular CaCl2 on tau protein levels in primary rat septo-hippocampal cultures. One day after injury, Western blot analyses revealed a calcium dependent loss of tau protein of approximately 50% of control values. Loss of tau protein was associated with calpain 1 mediated breakdown products to alpha-spectrin. Calpain inhibitors 1 and 2, applied immediately after depolarization injury and available to cultures for 24 h reduced depolarization induced degradation of tau protein to approximately 35% or 25% of control values, respectively. We propose that brief potassium depolarization causes degradation of tau protein, possibly due to calpain activation. Thus, calpain inhibitors could represent a viable strategy for preserving the cytoskeletal structure of injured neurons.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Blotting, Western
  • Calcium Chloride / pharmacology
  • Cells, Cultured / drug effects
  • Dose-Response Relationship, Drug
  • Glycoproteins / pharmacology*
  • Hippocampus / drug effects*
  • Hippocampus / metabolism
  • Potassium / pharmacology
  • Rats
  • Rats, Inbred Strains
  • Time Factors
  • tau Proteins / biosynthesis*
  • tau Proteins / drug effects*

Substances

  • Glycoproteins
  • calpain inhibitors
  • tau Proteins
  • Calcium Chloride
  • Potassium