Restoration of tumor oxygenation after cytotoxic therapy by a perflubron emulsion/carbogen breathing

Artif Cells Blood Substit Immobil Biotechnol. 1995;23(3):423-9. doi: 10.3109/10731199509117958.

Abstract

Female, Fisher 344 rats bearing 13762 mammary carcinoma implanted subcutaneously in a hind limb were treated with standard therapeutic single doses of antitumor treatments of several types including: 1) antitumor alkylating agents (cisplatin, cyclophosphamide); 2) natural products (adriamycin, taxol and etoposide); 3) antimetabolites (5-flourouracil); 4) hypoxic cell selective agents (mitomycin C, SR-4233) as well as 5) fractionated radiation therapy (3 Gray daily for 5 days). The oxygen levels in the tumors were measured in the absence of treatment and 24 hrs. after treatment using an Eppendorf p02 histograph. Fifty- to sixty-points were measured per tumor and 8-10 tumors comprised each group. The tumors were more hypoxic post treatment with every anticancer drug or radiation. The percent of p02 readings < or = 5 mmHg in the untreated tumors ranged from 85% (x-rays) to 59% (etoposide). Administration of the perflubron emulsion (8 ml/kg) and carbogen breathing (95% O2/5% CO2) increased the oxygenation of the tumors such that the percent of pO2 readings < or = 5 mmHg was 32% in the untreated controls and ranged from 27% (x-rays) to 56% (adria) in the treated tumors. These results indicate that administration of a perflubron emulsion/carbogen can increase the oxygen content of tumors when hypoxia is the result of cytotoxic therapy.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Antineoplastic Agents / therapeutic use*
  • Carbon Dioxide / therapeutic use*
  • Cell Hypoxia / drug effects
  • Cell Survival / drug effects
  • Combined Modality Therapy
  • Drug Synergism
  • Emulsions
  • Female
  • Fluorocarbons / therapeutic use*
  • Hydrocarbons, Brominated
  • Mammary Neoplasms, Experimental / drug therapy*
  • Mammary Neoplasms, Experimental / metabolism
  • Oxygen / metabolism*
  • Oxygen / therapeutic use*
  • Radiation-Sensitizing Agents / therapeutic use*
  • Rats
  • Rats, Inbred F344
  • Respiration

Substances

  • Antineoplastic Agents
  • Emulsions
  • Fluorocarbons
  • Hydrocarbons, Brominated
  • Radiation-Sensitizing Agents
  • Carbon Dioxide
  • carbogen
  • perflubron
  • Oxygen