Potassium single-channel properties in normal and Rous sarcoma virus-transformed chicken embryo fibroblasts

Pflugers Arch. 1994 May;427(1-2):17-23. doi: 10.1007/BF00585937.

Abstract

Ion channels in normal and Rous sarcoma virus (RSV)-transformed chicken embryo fibroblasts (CEFs) were examined by using the patch-clamp technique. Three different types of ion channels were observed with single-channel conductances in symmetrical 140 mM KCl (with frequencies of occurrence in parentheses) of 186 pS (70%), 110 pS (10%), and 65 pS (20%), which are identical in normal and RSV-transformed CEFs. The total channel density in both cell types is about 0.13 per micron2. All three types of channels are highly selective for K+ ions, they are Ca(2+)- and voltage-dependent, and they can be completely blocked by external tetraethylammonium (10 mM) in both normal and RSV-transformed cells. Some channel properties, however, are different in normal and RSV-transformed CEFs. The K186 channel of normal CEFs is almost completely activated in the presence of about 1 nM free internal Ca2+ and is insensitive to charybdotoxin (100 nM). In contrast, the K186 channel of RSV-transformed CEFs has an EC50 value for activation by internal Ca2+ of about 100 nM and is highly sensitive to charybdotoxin (IC50 = 9 nM). In normal CEFs, the K186 channel activity starts at membrane potentials more positive than -50 mV and reaches a high open state probability of 0.94 at +50 mV. In RSV-transformed CEFs, the threshold of K186 channel activity is also -50 mV but the maximal open state probability is only 0.70 at +50 mV membrane potential. Averages of current traces of K186 channels show the typical features of the macroscopic K+ currents described previously for normal and RSV-transformed CEFs.(ABSTRACT TRUNCATED AT 250 WORDS)

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Avian Sarcoma Viruses / physiology*
  • Calcium / pharmacology
  • Cell Line, Transformed / metabolism
  • Cell Transformation, Viral*
  • Charybdotoxin
  • Chick Embryo / cytology*
  • Chick Embryo / metabolism*
  • Electrophysiology
  • Fibroblasts / metabolism
  • Potassium / pharmacokinetics
  • Potassium Channel Blockers
  • Potassium Channels / classification
  • Potassium Channels / physiology*
  • Reference Values
  • Scorpion Venoms / pharmacology

Substances

  • Potassium Channel Blockers
  • Potassium Channels
  • Scorpion Venoms
  • Charybdotoxin
  • Potassium
  • Calcium