Bruton tyrosine kinase is tyrosine phosphorylated and activated in pre-B lymphocytes and receptor-ligated B cells

Proc Natl Acad Sci U S A. 1994 Oct 25;91(22):10606-9. doi: 10.1073/pnas.91.22.10606.

Abstract

The gene encoding Bruton tyrosine kinase (Btk) is known to be mutated in human X chromosome-linked agammaglobulinemia and in the Xid mouse. This kinase was examined in B lymphocytes before and after antigen receptor ligation and also in pre-B cells. Btk was found to be catalytically activated and tyrosine phosphorylated in response to anti-IgM stimulation in B cells. This kinase is also constitutively phosphorylated on tyrosine residues in pre-B cells. These findings point to a functional role for Btk in pre-antigen and antigen receptor signaling during B-cell development and provide a biochemical explanation for the X-linked genetic syndromes already linked to this kinase.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Agammaglobulinaemia Tyrosine Kinase
  • Agammaglobulinemia / genetics
  • Agammaglobulinemia / immunology
  • Animals
  • B-Lymphocytes / enzymology*
  • B-Lymphocytes / immunology
  • Cell Line
  • Enzyme Activation
  • Hematopoietic Stem Cells / enzymology
  • Hematopoietic Stem Cells / immunology
  • Humans
  • Immunoglobulin M
  • Kinetics
  • Mice
  • Mice, Mutant Strains
  • Models, Biological
  • Mutation
  • Phosphorylation
  • Phosphotyrosine
  • Protein-Tyrosine Kinases / isolation & purification
  • Protein-Tyrosine Kinases / metabolism*
  • Receptors, Antigen, T-Cell / metabolism*
  • Signal Transduction
  • Tyrosine / analogs & derivatives
  • Tyrosine / analysis
  • X Chromosome

Substances

  • Immunoglobulin M
  • Receptors, Antigen, T-Cell
  • Phosphotyrosine
  • Tyrosine
  • Protein-Tyrosine Kinases
  • Agammaglobulinaemia Tyrosine Kinase
  • BTK protein, human
  • Btk protein, mouse