Transforming growth factor-beta regulates human retinal pigment epithelial cell phagocytosis by influencing a protein kinase C-dependent pathway

Graefes Arch Clin Exp Ophthalmol. 1994 Nov;232(11):695-701. doi: 10.1007/BF00171387.

Abstract

Background: Transforming growth factor-beta (TGF-beta) plays an important role in the pathogenesis of many ocular diseases, including proliferative vitreoretinopathy. We examined the effect of TGF-beta on the phagocytosis of rod outer segments by retinal pigment epithelium (RPE), which is a major function of RPE, and investigated the dependence of this effect on the protein kinase C (PKC) pathway.

Methods: Phagocytotic uptake of fluoresceinated bovine rod outer segments was determined by flow cytometry. RPE cells were treated with TGF-beta 1 or TGF-beta 2 and their effects on phagocytosis were examined. The effects of various PKC inhibitors (calphostin C, staurosporine, and extended exposure to phorbol 12-myristate 13-acetate, PMA) and a stimulator (brief exposure to PMA) on RPE phagocytosis was evaluated.

Results: Both TGF-beta 1 and TGF-beta 2 up-regulated RPE phagocytosis and PMA abolished the up-regulating effect of TGF-beta. In contrast, PKC inhibition by staurosporine and calphostin C resulted in increased phagocytosis. A combination of TGF-beta and PKC inhibitor treatment did not produced any additive effect on phagocytosis.

Conclusion: We concluded that TGF-beta up-regulates human RPE phagocytosis, but that this effect is counteracted by PKC activation. It is possible that this TGF-beta-induced effect is due, in part, to a negative modulation of the PKC-dependent pathway.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Alkaloids / pharmacology
  • Animals
  • Cattle
  • Cells, Cultured
  • Flow Cytometry
  • Humans
  • Naphthalenes*
  • Phagocytosis / drug effects
  • Phagocytosis / physiology*
  • Pigment Epithelium of Eye / cytology
  • Pigment Epithelium of Eye / drug effects
  • Pigment Epithelium of Eye / metabolism*
  • Polycyclic Compounds / pharmacology
  • Protein Kinase C / antagonists & inhibitors
  • Protein Kinase C / metabolism*
  • Rod Cell Outer Segment / physiology
  • Staurosporine
  • Tetradecanoylphorbol Acetate / pharmacology
  • Transforming Growth Factor beta / pharmacology*
  • Up-Regulation / drug effects

Substances

  • Alkaloids
  • Naphthalenes
  • Polycyclic Compounds
  • Transforming Growth Factor beta
  • calphostin complex
  • Protein Kinase C
  • Staurosporine
  • Tetradecanoylphorbol Acetate