[The effect of nicorandil on the neuromuscular block induced by vecuronium]

Masui. 1995 Jul;44(7):986-9.
[Article in Japanese]

Abstract

The effect of nicorandil on the neuromuscular block induced by vecuronium was investigated in vitro with rat phrenic nerve-hemidiaphragm preparation. Both single twitch (ST) and train-of-four ratio (TOFR) elicited with indirect electrical stimulation were used. The administration of nicorandil alone showed no effects on ST and TOFR. The pre-administration of nicorandil exerted significant depressing effect on ST compared with vecuronium alone. High concentration of nicorandil (4 x 10(-6) M) produced more significant effect on ST compared with low concentration of nicorandil (10(-7) M). In this study, the nicorandil showed similar effect as calcium antagonists on neuromuscular blockade.

Publication types

  • English Abstract

MeSH terms

  • Animals
  • Electric Stimulation
  • Male
  • Neuromuscular Blocking Agents / pharmacology*
  • Niacinamide / analogs & derivatives*
  • Niacinamide / pharmacology
  • Nicorandil
  • Phrenic Nerve / drug effects
  • Rats
  • Vecuronium Bromide / pharmacology*

Substances

  • Neuromuscular Blocking Agents
  • Niacinamide
  • Nicorandil
  • Vecuronium Bromide