Cytogenetic effects of 3-chloro-4-(dichloromethyl)-5-hydroxy-2(5H)-furanone (MX) in rat peripheral lymphocytes in vitro and in vivo

Mutat Res. 1993 Mar;299(1):25-8. doi: 10.1016/0165-1218(93)90115-t.

Abstract

3-Chloro-4-(dichloromethyl)-5-hydroxy-2(5H)-furanone (MX) is a potent direct-acting Salmonella mutagen found in wood pulp chlorination effluents and chlorinated drinking water. In cultured rat peripheral lymphocytes, MX induced significant dose-related increases in sister-chromatid exchanges (SCEs) and chromosome aberrations at doses of 20-60 micrograms/ml and of 60-80 micrograms/ml, respectively. MX produced primarily chromatid-type as opposed to chromosome-type aberrations. The peripheral lymphocytes of male and female rats exposed to MX by gavage 5 days a week for 14-18 weeks showed significant dose-related increases in SCEs at both levels of exposure (30 and 45-75 mg/kg) in both sexes. The present results demonstrate for the first time that MX is genotoxic in vivo.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cells, Cultured
  • Chromosome Aberrations*
  • Female
  • Furans / toxicity*
  • Lymphocytes / drug effects
  • Male
  • Mutagens / toxicity*
  • Rats
  • Rats, Wistar
  • Sister Chromatid Exchange*

Substances

  • Furans
  • Mutagens
  • 3-chloro-4-(dichloromethyl)-5-hydroxy-2(5H)-furanone