Profound differences in potassium current properties of normal and Rous sarcoma virus-transformed chicken embryo fibroblasts

Proc Natl Acad Sci U S A. 1993 Apr 15;90(8):3403-7. doi: 10.1073/pnas.90.8.3403.

Abstract

The membrane currents of chicken embryo fibroblasts (CEFs) transformed by Rous sarcoma virus (RSV) were compared with the currents of their nontransformed counterparts by using the whole-cell patch-clamp technique. In nontransformed CEFs, the main membrane current is a delayed outward K+ current that is sensitive to tetraethylammonium ion but insensitive to 4-aminopyridine. This K+ current is almost independent of the intracellular Ca2+ concentration and becomes completely inactivated at positive membrane potentials with a time constant of about 10 s at +30 mV. In contrast, transformed CEFs exhibit a noninactivating K+ current that strongly depends on the intracellular Ca2+ concentration. This Ca(2+)-dependent K+ current is blocked by the scorpion toxin charybdotoxin with an IC50 value of 19 nM, whereas the K+ current of normal CEFs is insensitive to charybdotoxin (up to 300 nM). The K+ current properties of transformed CEFs were also found after microinjection of purified, enzymatically active pp60v-src into normal CEFs but not after infection of CEFs with the Rous-associated virus RAV5, which lacks the v-src oncogene. Our results suggest that the oncogene product pp60v-src modulates existing K+ channel proteins, leading to profound electrophysiological and pharmacological alterations of the K+ current properties in RSV-transformed CEFs. Furthermore, our experiments identify for the first time K+ channels as possible substrates of pp60v-src.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apamin / pharmacology
  • Avian Sarcoma Viruses / genetics*
  • Cell Transformation, Neoplastic*
  • Cells, Cultured
  • Charybdotoxin
  • Chick Embryo
  • Elapid Venoms / pharmacology
  • Fibroblasts / physiology
  • Kinetics
  • Membrane Potentials / drug effects
  • Microinjections
  • Oncogene Protein pp60(v-src) / administration & dosage
  • Oncogene Protein pp60(v-src) / metabolism*
  • Potassium Channels / drug effects
  • Potassium Channels / physiology*
  • Scorpion Venoms / pharmacology

Substances

  • Elapid Venoms
  • Potassium Channels
  • Scorpion Venoms
  • Charybdotoxin
  • Apamin
  • dendrotoxin
  • Oncogene Protein pp60(v-src)