Differential requirement of a motif within the carboxyl-terminal domain of alpha-platelet-derived growth factor (alpha PDGF) receptor for PDGF focus forming activity chemotaxis, or growth

J Biol Chem. 1995 Mar 31;270(13):7033-6. doi: 10.1074/jbc.270.13.7033.

Abstract

To determine the molecular basis for the transforming function of platelet-derived growth factor (PDGF)-A in NIH/3T3 cells, we have constructed chimerae consisting of the extracellular domain of the human CSF-1R (fms) linked to the cytoplasmic domain of the alpha PDGF receptor (alpha R) containing a series of deletion or point mutations. The ability of fms/alpha R chimerae to mediate CSF-1-dependent anchorage-independent growth, focus formation, and chemotaxis of NIH/3T3 cells was then examined. Our results provide evidence that a domain encompassing amino acid residues 977-1024 of the alpha PDGFR is required for ligand-dependent focus formation, but not chemotaxis or anchorage-independent growth, and that tyrosine residues within this domain constitute the major binding site for phospholipase C gamma. Therefore, our findings suggest that: (i) the focus forming function of alpha PDGFR correlates well with the ability of the receptor to bind phospholipase C gamma, and (ii) the mechanism of focus formation mediated by alpha PDGFR may be distinguished from that required for chemotaxis or anchorage-independent growth.

MeSH terms

  • 3T3 Cells
  • Animals
  • Binding Sites
  • Cell Division / drug effects
  • Cell Division / physiology
  • Chemotaxis / drug effects
  • Chemotaxis / physiology*
  • Humans
  • Macrophage Colony-Stimulating Factor / pharmacology
  • Mice
  • Mutagenesis, Site-Directed
  • Platelet-Derived Growth Factor / pharmacology
  • Point Mutation
  • Receptor, Macrophage Colony-Stimulating Factor / biosynthesis
  • Receptor, Macrophage Colony-Stimulating Factor / physiology*
  • Receptor, Platelet-Derived Growth Factor alpha
  • Receptors, Platelet-Derived Growth Factor / biosynthesis
  • Receptors, Platelet-Derived Growth Factor / physiology*
  • Recombinant Fusion Proteins / biosynthesis
  • Recombinant Fusion Proteins / metabolism
  • Recombinant Proteins / metabolism
  • Recombinant Proteins / pharmacology
  • Sequence Deletion
  • Transfection
  • Type C Phospholipases / metabolism

Substances

  • Platelet-Derived Growth Factor
  • Recombinant Fusion Proteins
  • Recombinant Proteins
  • Macrophage Colony-Stimulating Factor
  • Receptor, Macrophage Colony-Stimulating Factor
  • Receptor, Platelet-Derived Growth Factor alpha
  • Receptors, Platelet-Derived Growth Factor
  • Type C Phospholipases