In-vitro and in-vivo activity of a new quinolone AM-1155 against Mycoplasma pneumoniae

J Antimicrob Chemother. 1994 Dec;34(6):875-83. doi: 10.1093/jac/34.6.875.

Abstract

We investigated the in-vitro and in-vivo activity of a new quinolone AM-1155 against Mycoplasma pneumoniae, and compared it with ofloxacin, ciprofloxacin, lomefloxacin, tosufloxacin, erythromycin and minocycline. AM-1155 was the most potent agent in vitro of the quinolones tested. Its pre-treatment minimal inhibitory concentrations for 90% of the 41 strains (MIC90) was 0.06 mg/L. In contrast, pre-treatment MIC90 values for ofloxacin, ciprofloxacin, lomefloxacin, tosufloxacin, erythromycin, and minocycline were 1, 1, 2, 0.5, 0.0156, and 0.5 mg/L, respectively. Post-treatments MIC90s, which may reflect mycoplasmacidal potency, of AM-1155, ofloxacin, ciprofloxacin, lomefloxacin, tosufloxacin, erythromycin and minocycline were 0.125, 1, 2, 4, 0.5, 0.125 and 4 mg/L, respectively. In-vitro activities of antimicrobial agents were assessed in an experimental pulmonary infection model in Syrian golden hamsters. AM-1155 was the most effective agent among five antimicrobial agents (AM-1155, ofloxacin, tosufloxacin, erythromycin, minocycline) tested in terms of reduction in viable M. pneumoniae cells and in reducing macroscopic lung lesions. These results suggest that AM-1155 will be a useful antimicrobial agent for the treatment of M. pneumoniae infections.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Anti-Infective Agents / pharmacology
  • Cell Death / drug effects
  • Cricetinae
  • Disease Models, Animal
  • Erythromycin / pharmacology
  • Fluoroquinolones*
  • Gatifloxacin
  • Lung / chemistry
  • Male
  • Mesocricetus
  • Minocycline / pharmacology
  • Mycoplasma pneumoniae / drug effects*
  • Piperazines / analysis
  • Piperazines / pharmacology*
  • Pneumonia, Mycoplasma / drug therapy
  • Quinolones / analysis
  • Quinolones / pharmacology*

Substances

  • Anti-Infective Agents
  • Fluoroquinolones
  • Piperazines
  • Quinolones
  • Erythromycin
  • Minocycline
  • Gatifloxacin