Cross-tolerance to ethanol and gamma-hydroxybutyric acid

Eur J Pharmacol. 1995 Feb 6;273(3):235-8. doi: 10.1016/0014-2999(94)00687-3.

Abstract

In the present study, the development of tolerance to the motor impairing effects of gamma-hydroxybutyric acid (GHBA) and ethanol was compared (Experiment 1). Rats were required to perform a motor coordination task daily shortly after ethanol (3.5 g/kg) and GHBA (1.0 g/kg) administration for 9 consecutive days. Tolerance to the motor impairing effects of ethanol and GHBA developed to a similar extent but with different patterns. On the tenth day, the presence of cross-tolerance to the motor impairing effects of GHBA and ethanol was assessed (Experiment 2). Administration of 1.0 g/kg GHBA produced a significantly lower impairment in ethanol-tolerant rats than in ethanol-naive rats. Similarly, administration of 3.5 g/kg ethanol induced a significantly lower impairment in GHBA-tolerant rats than in GHBA-naive rats. The presence of cross-tolerance between GHBA and ethanol is discussed in terms of common pathways of neuroadaptation to chronic GHBA and ethanol.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Ataxia / chemically induced*
  • Ataxia / psychology
  • Dose-Response Relationship, Drug
  • Drug Tolerance
  • Ethanol / pharmacology*
  • Male
  • Postural Balance / drug effects
  • Rats
  • Rats, Sprague-Dawley
  • Sodium Oxybate / pharmacology*

Substances

  • Ethanol
  • Sodium Oxybate