Opening of brain potassium-channels inhibits the ACTH-induced behavioral syndrome in the male rat

Neurosci Lett. 1995 Mar 16;188(1):29-32. doi: 10.1016/0304-3940(95)11387-c.

Abstract

In adult male rats, the intracerebroventricular (i.c.v.) injection of pinacidil, a potassium channel opener, at the doses of 100, 200 or 300 micrograms/rat, dose-dependently reduced the display of the most typical behavioral symptoms (excessive grooming, stretching, yawning, penile erections) induced by the i.c.v. administration of ACTH-(1-24) (4 micrograms/rat). These data indicate that the complex mechanism of the melanocortin-induced behavioral syndrome involves closure of potassium channels in target neurons, and provide further experimental support to the idea that melanocortins are functional antagonists of opioids.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Behavior, Animal / drug effects*
  • Behavior, Animal / physiology
  • Cosyntropin / pharmacology*
  • Dimethyl Sulfoxide / pharmacology
  • Dose-Response Relationship, Drug
  • Grooming / drug effects
  • Grooming / physiology
  • Guanidines / cerebrospinal fluid
  • Guanidines / pharmacology*
  • Injections, Intraventricular
  • Male
  • Penile Erection / drug effects
  • Pinacidil
  • Potassium Channels / drug effects*
  • Potassium Channels / physiology
  • Rats
  • Rats, Wistar

Substances

  • Guanidines
  • Potassium Channels
  • Cosyntropin
  • Pinacidil
  • Dimethyl Sulfoxide