N-arginine dibasic convertase (NRD convertase): a newcomer to the family of processing endopeptidases. An overview

Biochimie. 1994;76(3-4):234-40. doi: 10.1016/0300-9084(94)90151-1.

Abstract

N-arginine dibasic convertase (NRD convertase) (accession number L27124) is a metalloendopeptidase from rat brain cortex and testis which cleaves peptide substrates on the N-terminus of arginine residues in basic doublets. Its predicted amino acid sequence contains the putative zinc binding motif HXXEH in a region which exhibits 35% and 48% similarity with E coli protease III (pitrilysin E.C 3.4.99.44) and rat or human insulinase (E.C 3.4.99.45) respectively. This feature clearly classifies this endopeptidase as a member of the pitrilysin family of zinc-metalloproteases. However, the NRD convertase sequence contains a distinctive additional feature consisting of a 71 acidic amino acid stretch. Its substrate selectivity and the characteristic motifs of its amino acid sequence allow us to propose this new metalloendopeptidase as the first member of a new class of processing enzymes.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Cerebral Cortex / enzymology*
  • Cloning, Molecular
  • Dynorphins / chemistry
  • Dynorphins / metabolism
  • Kinetics
  • Male
  • Metalloendopeptidases / chemistry
  • Metalloendopeptidases / isolation & purification
  • Metalloendopeptidases / metabolism*
  • Molecular Sequence Data
  • Organ Specificity
  • Peptide Fragments / chemistry
  • Peptide Fragments / metabolism
  • Rats
  • Recombinant Proteins / chemistry
  • Sequence Homology, Amino Acid
  • Somatostatin / chemistry
  • Somatostatin / metabolism
  • Substrate Specificity
  • Testis / enzymology*

Substances

  • Peptide Fragments
  • Recombinant Proteins
  • Somatostatin
  • Dynorphins
  • Metalloendopeptidases
  • nardilysin