Inhibition of the effects of TNF in renal allograft recipients using recombinant human dimeric tumor necrosis factor receptors

Transplantation. 1995 Jan 27;59(2):300-5.

Abstract

Tumor necrosis factor alpha (TNFa) and lymphotoxin (LT) or TNF beta are closely linked cytokines produced by macrophages and activated T lymphocytes, which play important regulatory roles in the immune response to allografts. They have also been implicated as mediators of the adverse reactions observed during OKT3 therapy. Therefore, anti-TNF agents could be useful both for immunosuppression and for limiting the systemic response observed in patients receiving OKT3. Recombinant TNFR:Fc is a fusion protein that binds TNFa and LT, thereby neutralizing their effects in vitro. The present study investigates the potential clinical application of TNFR:Fc in a nonhuman primate renal allograft model. Cynomolgus renal allograft recipients were treated with TNFR:Fc induction therapy alone or in combination with subtherapeutic doses of cyclosporine. Control animals received no immunosuppression or subtherapeutic cyclosporine. TNFR:Fc, administered as the only immunosuppressive agent, successfully prolonged renal allograft survival in the majority of treated animals. The prolongation of allograft survival was even more impressive when TNFR:Fc was combined with subtherapeutic doses of cyclosporine. Onset of rejection was significantly delayed as well in the TNFR:Fc treated groups. No adverse side effects were observed in any of the TNFR:Fc treated animals. Precursor cytotoxic T cells were detected in peripheral blood samples of treated recipients but the level of effector CTLs in vivo was below the threshold of detection. These results demonstrate that TNFR:Fc can be safely administered and is effective in prolonging renal allograft survival and in delaying the onset of rejection when administered alone or in combination with cyclosporine.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Graft Survival / drug effects
  • Immunity, Cellular / drug effects
  • Immunoglobulin Fc Fragments / pharmacology
  • Immunosuppressive Agents / pharmacology*
  • Immunotoxins / pharmacology*
  • Kidney Transplantation / immunology*
  • Macaca fascicularis
  • Male
  • Models, Biological
  • Receptors, Tumor Necrosis Factor / physiology*
  • Recombinant Fusion Proteins / pharmacology
  • Recombinant Proteins / pharmacology
  • Solubility
  • Transplantation, Homologous
  • Tumor Necrosis Factor-alpha / antagonists & inhibitors*

Substances

  • Immunoglobulin Fc Fragments
  • Immunosuppressive Agents
  • Immunotoxins
  • Receptors, Tumor Necrosis Factor
  • Recombinant Fusion Proteins
  • Recombinant Proteins
  • Tumor Necrosis Factor-alpha