Effects of R80122, a new phosphodiesterase inhibitor, on liver and global haemodynamics in patients undergoing coronary artery bypass surgery

Cardiovasc Surg. 1994 Dec;2(6):698-702.

Abstract

R80122 (0.3 mg/kg body weight), a new phosphodiesterase inhibitor, was tested in ten patients undergoing coronary artery bypass surgery. Haemodynamic measurements were made and hepatic blood flow assessed by the indocyanine green infusion method using liver vein catheterization. Cardiac index increased by 63% and systemic vascular resistance decreased by 47%. Hepatic blood flow and intestinal vascular resistance were not significantly affected; nor was hepatic oxygen consumption. It is concluded that R80122 is a highly cardioselective phosphodiesterase inhibitor and that the reduction in systemic vascular resistance by this drug is not an effect of extensive intestinal vasodilatation.

Publication types

  • Clinical Trial

MeSH terms

  • Adult
  • Aged
  • Cardiotonic Agents / pharmacology*
  • Cardiotonic Agents / therapeutic use
  • Coronary Artery Bypass*
  • Coronary Disease / physiopathology
  • Coronary Disease / surgery
  • Hemodynamics / drug effects*
  • Humans
  • Imidazoles / pharmacology*
  • Imidazoles / therapeutic use
  • Intraoperative Care*
  • Liver / drug effects*
  • Liver / physiopathology
  • Male
  • Middle Aged
  • Phosphodiesterase Inhibitors / pharmacology*
  • Phosphodiesterase Inhibitors / therapeutic use
  • Quinazolines / pharmacology*
  • Quinazolines / therapeutic use
  • Statistics, Nonparametric

Substances

  • Cardiotonic Agents
  • Imidazoles
  • Phosphodiesterase Inhibitors
  • Quinazolines
  • R 80122