Synthesis of imidazo[2,1-b]thiazoles and thiazolines as potential antiulcer agents

J Pharm Belg. 1994 Jul-Aug;49(4):308-14.

Abstract

The replacement of the imidazole ring of cimetidine with a bicyclic system (imidazo[1,2-a]pyridine), reported in the literature, produced compounds endowed with potent antiulcer activity. In this paper we describe the synthesis of imidazo [2,1-b]thiazoles and thiazolines bearing the side chain of metiamide, cimetidine and ranitidine: the compounds obtained, tested on gastric lesions induced in rats by ethanol and by stress, were devoid of antiulcer activity.

MeSH terms

  • Animals
  • Anti-Ulcer Agents / chemical synthesis*
  • Anti-Ulcer Agents / pharmacology
  • Imidazoles / chemical synthesis*
  • Imidazoles / pharmacology
  • Peptic Ulcer Hemorrhage / etiology
  • Peptic Ulcer Hemorrhage / prevention & control
  • Rats
  • Stomach Ulcer / chemically induced
  • Stomach Ulcer / prevention & control
  • Thiazoles / chemical synthesis*
  • Thiazoles / pharmacology

Substances

  • Anti-Ulcer Agents
  • Imidazoles
  • Thiazoles