Solid state investigation of mefloquine hydrochloride

J Pharm Biomed Anal. 1994 Jul;12(7):889-93. doi: 10.1016/0731-7085(93)e0034-k.

Abstract

Mefloquine hydrochloride was crystallized under different conditions and the products were studied by thermal analysis, IR spectroscopy and X-ray diffraction. It was demonstrated that different conditions of crystallization resulted in different crystal structures. The alpha- and delta-modifications were hydrates, the beta- and gamma-forms were polymorphs, the epsilon-form was an acetone solvate and theta-mefloquine was tetrahydrofuran solvate. During long storage at room temperature, the alpha-, delta- and theta-forms of mefloquine hydrochloride were transformed. By heat treatment of the delta-, epsilon and theta-modifications, a new crystal structure was obtained.

MeSH terms

  • Calorimetry, Differential Scanning
  • Chromatography, Gas
  • Crystallography, X-Ray
  • Differential Thermal Analysis
  • Mefloquine / chemistry*
  • Spectrophotometry, Infrared
  • Thermogravimetry

Substances

  • Mefloquine