Disruption by interferon-alpha of an autocrine interleukin-6 growth loop in IL-6-dependent U266 myeloma cells by homologous and heterologous down-regulation of the IL-6 receptor alpha- and beta-chains

J Clin Invest. 1994 Dec;94(6):2317-25. doi: 10.1172/JCI117596.

Abstract

IL-6 is an autocrine growth factor for U266 myeloma cells and their growth is inhibited by IFN-alpha or IL-6 mAb. We asked, therefore, whether IFN-alpha-induced growth inhibition involved IL-6. IFN-alpha and mAb against IL-6, the IL-6R alpha-(gp80) or beta-chain (gp130) potently inhibited U266 cells. Remarkably, this effect occurred despite IFN-alpha-augmented secretion of endogenous IL-6. However, examining the IL-6R revealed that IFN-alpha drastically curtailed expression of the IL-6R alpha- and beta-chain. This effect occurred on two different levels (protein and mRNA) and by two different mechanisms (directly and indirectly through IL-6). First, IFN-alpha, but not IL-6, greatly decreased gp80 and, to a lesser extent, gp130 mRNA levels which resulted in a loss of IL-6 binding sites. Second, IFN-alpha-induced IL-6 predominantly down-regulated membrane-bound gp130. IFN-alpha-mediated decrease of gp80 levels was not detected on IL-6-independent myeloma (RPMI 8226) or myeloid cells (U937). We conclude that IFN-alpha inhibited IL-6-dependent myeloma cell growth by depriving U266 cells of an essential component of their autocrine growth loop, a functional IL-6R.

MeSH terms

  • Affinity Labels
  • Cell Division / drug effects
  • Cross-Linking Reagents
  • Cytokines / pharmacology
  • Dose-Response Relationship, Drug
  • Down-Regulation*
  • Humans
  • Interferon-alpha / pharmacology*
  • Interleukin-6 / pharmacology*
  • Multiple Myeloma / metabolism*
  • Receptors, Interleukin / biosynthesis*
  • Receptors, Interleukin / genetics
  • Receptors, Interleukin-6
  • Tumor Cells, Cultured

Substances

  • Affinity Labels
  • Cross-Linking Reagents
  • Cytokines
  • Interferon-alpha
  • Interleukin-6
  • Receptors, Interleukin
  • Receptors, Interleukin-6