Induction of WAF1/CIP1 by a p53-independent pathway

Cancer Res. 1994 Jul 1;54(13):3391-5.

Abstract

The p53-inducible gene WAF1/CIP1 encodes a M(r) 21,000 protein (p21) that has been shown to arrest cell growth by inhibition of cyclin-dependent kinases. Induction of WAF1/CIP1 in cells undergoing p53-dependent G1 arrest or apoptosis supports the idea that WAF1/CIP1 is a critical downstream effector of p53. In the present study, we used embryonic fibroblasts from p53 "knock-out" mice to demonstrate p53-independent induction of WAF1/CIP1. We show that serum or individual growth factors such as platelet-derived growth factor, fibroblast growth factor, and epidermal growth factor but not insulin are able to induce WAF1/CIP1 in quiescent p53-deficient cells as well as in normal cells. The kinetics of this transient induction, which is enhanced by cycloheximide, demonstrates that WAF1/CIP1 is an immediate-early gene the transcript of which reaches a peak at approximately 2 h following serum or growth factor stimulation. On the other hand, DNA damage elicited by gamma-irradiation induces WAF1/CIP1 in normal human and mouse fibroblasts but does not affect WAF1/CIP1 expression in p53-deficient cells. These results suggest the existence of two separate pathways for the induction of WAF1/CIP1, a p53-dependent one activated by DNA damage and a p53-independent one activated by mitogens at the entry into the cell cycle. The possible function of p21 at this early stage is discussed.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 3T3 Cells
  • Animals
  • Base Sequence
  • Cycloheximide / pharmacology
  • G1 Phase / genetics*
  • Gene Expression Regulation / physiology*
  • Genes, Immediate-Early / drug effects
  • Genes, Immediate-Early / physiology*
  • Genes, Immediate-Early / radiation effects
  • Genes, Tumor Suppressor / drug effects
  • Genes, Tumor Suppressor / physiology*
  • Genes, Tumor Suppressor / radiation effects
  • Genes, p53 / drug effects
  • Genes, p53 / physiology
  • Genes, p53 / radiation effects
  • Growth Substances / pharmacology
  • Insulin / pharmacology
  • Mice
  • Molecular Sequence Data
  • Platelet-Derived Growth Factor / pharmacology
  • Tumor Cells, Cultured
  • Tumor Suppressor Protein p53 / deficiency

Substances

  • Growth Substances
  • Insulin
  • Platelet-Derived Growth Factor
  • Tumor Suppressor Protein p53
  • Cycloheximide