Insulin-like effects of sodium orthovanadate on diacylglycerol-protein kinase C signaling in BC3H-1 myocytes

Arch Biochem Biophys. 1994 Jul;312(1):167-72. doi: 10.1006/abbi.1994.1295.

Abstract

In this paper we examine whether sodium orthovanadate activates diacylglycerol (DAG)/protein kinase C (PKC) signaling systems that are activated by insulin in BC3H-1 myocytes. Like insulin, sodium orthovanadate provoked increases in membrane DAG, PKC enzyme activity, and immunoreactive PKC-beta. Concomitantly, both PKC enzyme activity and immunoreactive PKC-beta decreased in the cytosol, suggesting that sodium orthovanadate, like insulin, stimulated the translocation of PKC-beta from the cytosol to the membrane fraction. Sodium orthovanadate was also found to activate phospholipid signaling pathways that were previously reported to be activated by insulin, viz., inositol-lipid synthesis/turnover; phosphatidylcholine hydrolysis; and de novo phospholipid synthesis by activation of glycerol-3-PO4 acyltransferase. Our findings suggest that vanadate mimics insulin in the activation of specific phospholipid/DAG/PKC signaling pathways.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Biological Transport
  • Cell Fractionation
  • Cytosol / enzymology
  • Diglycerides / metabolism*
  • Enzyme Activation
  • Glycerol-3-Phosphate O-Acyltransferase / metabolism
  • Insulin / pharmacology*
  • Isoenzymes / metabolism
  • Membranes / enzymology
  • Mice
  • Muscles / drug effects*
  • Phospholipids / metabolism
  • Protein Kinase C / metabolism*
  • Signal Transduction*
  • Vanadates / pharmacology*

Substances

  • Diglycerides
  • Insulin
  • Isoenzymes
  • Phospholipids
  • Vanadates
  • Glycerol-3-Phosphate O-Acyltransferase
  • Protein Kinase C