Transcriptional activation by the v-Jun oncoprotein is independent of positive regulatory phosphorylation

Oncogene. 1994 Aug;9(8):2363-8.

Abstract

Growth factors, phorbol esters, and oncogenes such as ras, src, and sis are believed to stimulate c-Jun transcriptional activation by inducing increased phosphorylation at two serine residues (S63 and S73) within the N-terminal transactivation domain. Although S63 and S73 are conserved in the mutant v-Jun oncoprotein, they are not phosphorylated by two enzymes which target the corresponding residues in c-Jun in vitro; namely a partially purified c-Jun kinase from TPA-stimulated U937 cells and purified p54 mitogen activated protein (MAP) kinase. In addition, v-Jun activates transcription more strongly than c-Jun when fused to the Gal4 DNA-binding domain, and transcriptional activation by Gal4-v-Jun is unaffected when S63, S73, or both, are replaced with non-phosphorylatable alanine residues, amino acid substitutions which severely impair transcriptional activation by Gal4-c-Jun. The novel biochemical and transcriptional properties of v-Jun result from deletion of a 27 amino acid segment, termed delta, which is important for transforming activity. On the basis of these results we propose that unlike c-Jun, v-Jun transcriptional activation is independent of positive regulatory phosphorylation and that this may contribute to oncogenesis by v-Jun.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Calcium-Calmodulin-Dependent Protein Kinases / metabolism
  • Chick Embryo
  • Humans
  • Oncogene Protein p65(gag-jun) / chemistry
  • Oncogene Protein p65(gag-jun) / physiology*
  • Phosphorylation
  • Proto-Oncogene Proteins c-jun / physiology
  • Structure-Activity Relationship
  • Transcriptional Activation*

Substances

  • Oncogene Protein p65(gag-jun)
  • Proto-Oncogene Proteins c-jun
  • Calcium-Calmodulin-Dependent Protein Kinases