Role of calcium in the bombesin-induced intestinal CCK release in rats

Peptides. 1993 Nov-Dec;14(6):1295-7. doi: 10.1016/0196-9781(93)90189-n.

Abstract

In the isolated vascularly perfused rat duodenojejunum, vascular infusion of bombesin (100 nM) provoked an early, transient (6 min) release of CCK (500% of basal), followed by a sustained response (400% of basal). The calcium chelator EGTA (2 mM) reduced the early peak and abolished the second phase of CCK release. A similar variation was evoked by verapamil (10 microM), whereas diltiazem (100 microM), nifedipine (50 microM), and omega-conotoxin (100 nM) had no significant effect. It is concluded that bombesin-induced CCK release from rat intestine is dependent on the availability of extracellular calcium and on the activation of calcium channels sensitive to blockers of the phenylalkylamine family.

MeSH terms

  • Animals
  • Bombesin / pharmacology*
  • Calcium / physiology*
  • Calcium Channel Blockers / pharmacology
  • Cholecystokinin / metabolism*
  • Diltiazem / pharmacology
  • In Vitro Techniques
  • Intestine, Small / drug effects*
  • Intestine, Small / metabolism
  • Male
  • Nifedipine / pharmacology
  • Peptides / pharmacology
  • Rats
  • Rats, Wistar
  • Verapamil / pharmacology
  • omega-Conotoxins*

Substances

  • Calcium Channel Blockers
  • Peptides
  • omega-Conotoxins
  • Conus magus toxin
  • Cholecystokinin
  • Verapamil
  • Diltiazem
  • Nifedipine
  • Bombesin
  • Calcium