Efficacy of 4-methylpyrazole in ethylene glycol poisoning: clinical and toxicokinetic aspects

Hum Exp Toxicol. 1994 Jan;13(1):61-4. doi: 10.1177/096032719401300109.

Abstract

Potentially fatal ethylene glycol intoxication in an adult with normal renal function was treated with 4-methylpyrazole administered three hours after the incident occurred. The plasma ethylene glycol concentration was 3.5 g l-1 on admission. The metabolic acidosis present on admission resolved within four hours, and the subsequent clinical course was uneventful. The apparent plasma half-life of ethylene glycol was 16 h and the mean renal and plasma clearances of ethylene glycol were 24 and 25 ml min-1, respectively. These results support the hypothesis that complete blockade of hepatic metabolism of ethylene glycol is achieved by 4-methylpyrazole. The only side-effect observed as a result of treatment was a transient slight increase in serum transaminase activity.

Publication types

  • Case Reports

MeSH terms

  • Adult
  • Ethylene Glycol
  • Ethylene Glycols / blood
  • Ethylene Glycols / poisoning*
  • Fomepizole
  • Humans
  • Male
  • Poisoning / drug therapy
  • Pyrazoles / therapeutic use*

Substances

  • Ethylene Glycols
  • Pyrazoles
  • Fomepizole
  • Ethylene Glycol