cDNA transfection followed by the isolation of a MCF-7 breast cell line resistant to tamoxifen in vitro and in vivo

Br J Cancer. 1993 Dec;68(6):1088-96. doi: 10.1038/bjc.1993.486.

Abstract

A tamoxifen resistant cell line (clone 9) has been isolated from the tamoxifen sensitive, hormone responsive MCF-7 breast carcinoma cell line after transfection with mixed cDNA libraries, followed by tamoxifen selection in the presence of oestrogens. Transfection was confirmed by Southern analysis with vector probes. Clone 9 in several-fold more resistant to tamoxifen and other anti-oestrogens than wild type cells when cultured either as a monolayer or as colonies in soft agar but retains oestrogen receptors. Clone 9 was less responsive to 17-beta-oestradiol than were wild type MCF-7. In addition to showing in vitro tamoxifen resistance, clone 9 was also tamoxifen resistant in vivo when xenografted into the nude mouse. Culture medium conditioned by clone 9 cells stimulated quiescent cells of the same clone as well as wild type cells, whereas medium conditioned by wild type MCF-7 was inhibitory to both, suggesting that clone 9 may be secreting an autocrine growth factor. Clone 9 provides a novel model for further investigation of the mechanism of anti-oestrogen resistance that occurs without loss of oestrogen receptors. Preliminary results suggest that an autocrine growth stimulatory mechanism may be one pathway of such resistance.

MeSH terms

  • Animals
  • Breast Neoplasms / drug therapy
  • Breast Neoplasms / genetics*
  • Cloning, Molecular
  • Culture Media, Conditioned
  • DNA, Complementary
  • DNA, Neoplasm / genetics*
  • DNA, Recombinant
  • Drug Resistance / genetics*
  • Estradiol / analogs & derivatives
  • Estradiol / pharmacology
  • Estrogen Antagonists / metabolism
  • Estrogens / metabolism
  • Female
  • Growth Substances / physiology
  • Humans
  • Mice
  • Mice, Inbred BALB C
  • Mice, Nude
  • Neoplasm Transplantation
  • Polyunsaturated Alkamides
  • Receptors, Estrogen / metabolism
  • Tamoxifen / analogs & derivatives
  • Tamoxifen / pharmacology*
  • Tamoxifen / therapeutic use
  • Transfection
  • Tumor Cells, Cultured / drug effects
  • Tumor Cells, Cultured / metabolism
  • Tumor Stem Cell Assay

Substances

  • Culture Media, Conditioned
  • DNA, Complementary
  • DNA, Neoplasm
  • DNA, Recombinant
  • Estrogen Antagonists
  • Estrogens
  • Growth Substances
  • Polyunsaturated Alkamides
  • Receptors, Estrogen
  • Tamoxifen
  • afimoxifene
  • Estradiol
  • ICI 164384