Chemical synthesis and biological activity of a novel antibacterial peptide deduced from a pig myeloid cDNA

FEBS Lett. 1994 Jan 17;337(3):303-7. doi: 10.1016/0014-5793(94)80214-9.

Abstract

Several myeloid precursors of antibacterial peptides have recently been shown to share homologous pre- and pro-regions. Taking advantage of this homology, a novel cDNA was cloned from pig bone marrow RNA. This encodes a 166-residue polypeptide with highly conserved pre- (29 residues) and pro- (101 residues) sequences, followed by a unique, 36-residue C-terminal sequence. Structure analyses of this C-terminal region have identified a highly cationic sequence predicted to adopt an amphipathic alpha-helical conformation. A peptide corresponding to this sequence was chemically synthesized and shown to arrest the growth of both Gram-positive and Gram-negative bacteria. At least for Escherichia coli, the activity of this peptide appears to be mediated by its ability to permeabilize the bacterial membranes.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Antimicrobial Cationic Peptides
  • Bacteria / drug effects*
  • Base Sequence
  • Bone Marrow / chemistry*
  • Cell Membrane Permeability / drug effects
  • Chromatography, High Pressure Liquid
  • Circular Dichroism
  • DNA, Complementary / chemistry*
  • DNA, Complementary / genetics
  • DNA, Complementary / isolation & purification
  • Escherichia coli / drug effects
  • Mass Spectrometry
  • Molecular Sequence Data
  • Peptides / chemical synthesis*
  • Peptides / genetics
  • Peptides / pharmacology
  • Polymerase Chain Reaction
  • Protein Structure, Secondary
  • Proteins / chemical synthesis*
  • Proteins / genetics
  • Proteins / pharmacology
  • Swine

Substances

  • Antimicrobial Cationic Peptides
  • DNA, Complementary
  • PMAP-36
  • Peptides
  • Proteins

Associated data

  • GENBANK/L29125