Effects of imidazole-salicylate on renal function and the diuretic action of furosemide in cirrhotic patients with ascites

J Hepatol. 1993 Sep;19(2):279-84. doi: 10.1016/s0168-8278(05)80583-5.

Abstract

Imidazole-salicylate is a non-steroidal anti-inflammatory drug with limited inhibitory effects on prostaglandin synthesis. The renal effects of this drug were investigated by a double-blind cross-over study in 10 patients with cirrhosis and ascites. Two therapeutic doses of imidazole-salicylate (750 mg each) were given at midnight and 08:00 h and 80 mg of furosemide were injected intravenously at 09:00 h. The same procedure was followed on another day but a placebo replaced imidazole-salicylate. Renal function (creatinine clearance, free water and electrolyte excretions) and urinary excretion of prostaglandin E, 6-keto-prostaglandin F1 alpha and thromboxane B2 were evaluated for 8 h after the first dose of the drug and for 2 h after furosemide injection. Platelet thromboxane production was also determined 9 h after the first administration of drug or placebo. Imidazole-salicylate did not affect renal function or inhibit kidney prostanoid production either under basal conditions or after the stimulating effect of furosemide. On the contrary, imidazole-salicylate significantly inhibited platelet thromboxane production (45.8 +/- 9 vs. 69.4 +/- 7.5 ng/ml, P < 0.05). These results suggest that imidazole-salicylate is an anti-inflammatory drug that can be given to patients with decompensated cirrhosis without risk of inhibiting kidney prostaglandin synthesis or the renal response to furosemide.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial

MeSH terms

  • Adult
  • Aged
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology*
  • Anti-Inflammatory Agents, Non-Steroidal / therapeutic use
  • Ascites / drug therapy
  • Ascites / metabolism
  • Ascites / physiopathology*
  • Blood Platelets / metabolism
  • Diuretics / pharmacology*
  • Diuretics / therapeutic use
  • Double-Blind Method
  • Female
  • Furosemide / pharmacology*
  • Furosemide / therapeutic use
  • Glomerular Filtration Rate / drug effects
  • Humans
  • Imidazoles / pharmacology*
  • Imidazoles / therapeutic use
  • Kidney / drug effects
  • Kidney / physiology*
  • Liver Cirrhosis / drug therapy
  • Liver Cirrhosis / metabolism
  • Liver Cirrhosis / physiopathology*
  • Male
  • Middle Aged
  • Prostaglandins F / urine
  • Salicylates / pharmacology*
  • Salicylates / therapeutic use
  • Thromboxane B2 / metabolism
  • Thromboxane B2 / urine
  • Time Factors

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Diuretics
  • Imidazoles
  • Prostaglandins F
  • Salicylates
  • imidazole-2-hydroxybenzoate
  • Thromboxane B2
  • Furosemide
  • prostaglandin F1