Chemical and biological properties of porcine secretin and secretin analogues modified in positions 3 and 4

Gastroenterology. 1977 Apr;72(4 Pt.2):797-800.

Abstract

The synthesis of secretin does not offer fundamental difficulties any longer. The problem of the stability of the hormone seems to be solved from a practical point of view. However, the mechanism of the inactivation of secretin in solution is not yet satisfactorily explained, alpha-beta Rearrangement of the Asp-Gly bond may play a role, but some observations indicate that inactivation is not a straight reaction. Like secretion [Ala-4] secretin shows beta-sympathomimetic activity. The availability of a suitable depot preparation permits physiological studies with secretin and its analogues after subcutaneous administration.

MeSH terms

  • Animals
  • Chemical Phenomena
  • Chemistry
  • Secretin* / analogs & derivatives*
  • Secretin* / chemical synthesis
  • Secretin* / isolation & purification
  • Swine

Substances

  • Secretin