Src homology 2 domains of protein tyrosine phosphatase are phosphorylated by insulin receptor kinase and bind to the COOH-terminus of insulin receptors in vitro

Biochem Biophys Res Commun. 1993 Jul 15;194(1):208-14. doi: 10.1006/bbrc.1993.1805.

Abstract

To clarify the role of protein tyrosine phosphatases(PTPase) containing Src homology 2 (SH2) regions on insulin signaling, we investigated the interactions between SH2 regions of PTPase and insulin receptors. We made a pair of SH2 domains of PTP1C and SH-PTP2 fusion proteins coupled to glutathione-S-transferase (GST) using pGEX-3X expression vector. After incubating with insulin, insulin receptors were incubated with SH2 proteins in the presence of 100 mu ATP at 4 degrees C for 3 hr, and then immunoprecipitated and analyzed by SDS-PAGE. We found that SH2 domains of SH-PTP2 were phosphorylated, but not those of PTP1C by insulin receptor kinase and the SH2 domains of SH-PTP2, but not those of PTP1C, directly bound to the phosphorylated COOH-terminus of insulin receptors in vitro.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Binding Sites
  • Cell Line
  • Cloning, Molecular
  • Glutathione Transferase / metabolism
  • Humans
  • Molecular Sequence Data
  • Phosphorylation
  • Polymerase Chain Reaction
  • Protein Tyrosine Phosphatases / metabolism*
  • Protein-Tyrosine Kinases / metabolism*
  • Receptor, Insulin / metabolism
  • Recombinant Fusion Proteins / metabolism
  • Restriction Mapping
  • Sequence Homology, Amino Acid
  • Signal Transduction
  • Substrate Specificity

Substances

  • Recombinant Fusion Proteins
  • Glutathione Transferase
  • Protein-Tyrosine Kinases
  • Receptor, Insulin
  • Protein Tyrosine Phosphatases