IBZM-SPECT as predictor for dopamimetic responsiveness of patients with de novo parkinsonian syndrome

Adv Neurol. 1993:60:519-24.

Abstract

IBZM-SPECT is useful as a predictor for the responsiveness to oral L-DOPA therapy in de novo parkinsonian patients. A reduction of postsynaptic dopamine D2 receptors in de novo parkinsonian patients makes the diagnosis of Parkinson's disease rather unlikely. Normal IBZM binding does not prove the diagnosis of Parkinson's disease; however, together with a positive apomorphine test, it strongly supports the clinical diagnosis. At present the combination of IBZM-SPECT and apomorphine testing appears to be a useful procedure for selecting de novo patients for clinical trials with new anti-parkinsonian therapy.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Oral
  • Adult
  • Aged
  • Aged, 80 and over
  • Apomorphine*
  • Benzamides / pharmacokinetics*
  • Corpus Striatum / diagnostic imaging
  • Corpus Striatum / drug effects
  • Dopamine D2 Receptor Antagonists*
  • Female
  • Humans
  • Levodopa / therapeutic use*
  • Male
  • Middle Aged
  • Parkinson Disease / diagnostic imaging*
  • Parkinson Disease / drug therapy
  • Prospective Studies
  • Pyrrolidines / pharmacokinetics*
  • Receptors, Dopamine D1 / drug effects
  • Receptors, Dopamine D1 / physiology
  • Receptors, Dopamine D2 / physiology
  • Tomography, Emission-Computed, Single-Photon*

Substances

  • Benzamides
  • Dopamine D2 Receptor Antagonists
  • Pyrrolidines
  • Receptors, Dopamine D1
  • Receptors, Dopamine D2
  • Levodopa
  • 3-iodo-2-hydroxy-6-methoxy-N-((1-ethyl-2-pyrrolidinyl)methyl)benzamide
  • Apomorphine