Identification and characterization of an anti-tyrosine kinase factor in cystic gliomas

FEBS Lett. 1993 Jan 25;316(2):147-51. doi: 10.1016/0014-5793(93)81204-d.

Abstract

In view of the frequent activation of the epidermal growth factor receptor (EGF-R) in gliomas and autocrine hypothesis, we searched for 'EGF-like' factor(s) in cystic fluids (CFs) associated with gliomas. Membranes of A431 cells, which overexpress EGF-R, were used to explore such activity in 20 CFs. In all cases CFs induced inhibition of EGF-R phosphorylation. Biochemical analysis revealed an anti-tyrosine kinase activity which was identified as a 18 kDa proteic factor. Effectiveness at high dilution and anti-proliferative effect on living cells in culture suggest that this factor may be involved in the negative regulation of glial oncogenesis.

MeSH terms

  • Astrocytoma / chemistry*
  • Brain Neoplasms / chemistry*
  • Chromatography, High Pressure Liquid
  • Electrophoresis, Polyacrylamide Gel
  • ErbB Receptors / metabolism
  • Humans
  • Phosphorylation
  • Protein-Tyrosine Kinases / antagonists & inhibitors*
  • Tumor Cells, Cultured

Substances

  • ErbB Receptors
  • Protein-Tyrosine Kinases