Effect of oxymetazoline on nasal and sinus mucosal blood flow in the rabbit as measured with laser-Doppler flowmetry

Ann Otol Rhinol Laryngol. 1993 Feb;102(2):123-6. doi: 10.1177/000348949310200209.

Abstract

The effect of topical oxymetazoline hydrochloride on the blood flow of the nasal and sinus mucosa of the rabbit was measured by laser-Doppler flowmetry. Oxymetazoline, the active component in clinically used nose drops, induced a dose-dependent decrease of the nasal mucosal blood flow. This effect has previously been shown in humans and suggests the presence of alpha 2-adrenoceptors in the nasal mucosa of the rabbit. Doses of oxymetazoline used clinically in humans induced a 50% reduction of blood flow in rabbits. Rhythmic variations in blood flow were seen in 30% of the rabbits after administration of oxymetazoline. Additionally, oxymetazoline induced a dose-dependent decrease of the mucosal blood flow in the maxillary sinus when the drug was applied in the nose. A vasoconstricting effect of oxymetazoline on the arteries penetrating the maxillary sinus ostium is a possible explanation. This can have positive as well as negative consequences on acute sinus infections.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Administration, Intranasal
  • Animals
  • Dose-Response Relationship, Drug
  • Humans
  • Laser-Doppler Flowmetry
  • Male
  • Maxillary Sinus / blood supply*
  • Mucous Membrane / blood supply
  • Nasal Mucosa / blood supply*
  • Oxymetazoline / administration & dosage
  • Oxymetazoline / pharmacology*
  • Rabbits
  • Regional Blood Flow / drug effects

Substances

  • Oxymetazoline