Construction of synthetic signals for glycosyl-phosphatidylinositol anchor attachment. Analysis of amino acid sequence requirements for anchoring

J Biol Chem. 1993 Mar 25;268(9):6689-93.

Abstract

Many membrane proteins are anchored to the cell surface through covalent attachment to a glycosyl-phosphatidylinositol (GPI) structure. The GPI anchor is added to proteins in the endoplasmic reticulum following recognition of a signal in the COOH terminus of the protein. We show that the GPI anchoring signal can be completely recreated by the synthetic polymer Ser3-Thr8-Leu14, but not Thr11-Leu14, inserted at the COOH terminus of a protein. This is consistent with previous reports that a small amino acid such as Ser, Gly, or Ala, but not Thr, is required at the GPI attachment site. Analysis of synthetic amino acid sequences established a basic three-part signal for GPI anchoring: a cleavage/attachment domain that requires small amino acids at the first (GPI anchor attachment) and third positions but with little specificity at the middle position, a spacer domain of approximately 8-12 amino acids, and a hydrophobic domain of at least 11 amino acids. The ability to design a totally synthetic GPI anchoring signal will allow precise probing of the fine structure of this signal.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Amino Acids / metabolism
  • Animals
  • Antigens, CD / metabolism
  • CHO Cells
  • Cloning, Molecular
  • Cricetinae
  • Glycosylphosphatidylinositols / metabolism*
  • Humans
  • Membrane Cofactor Protein
  • Membrane Glycoproteins / metabolism
  • Mice
  • Molecular Sequence Data
  • Protein Sorting Signals / chemical synthesis
  • Protein Sorting Signals / metabolism*

Substances

  • Amino Acids
  • Antigens, CD
  • CD46 protein, human
  • Glycosylphosphatidylinositols
  • Mcp protein, mouse
  • Membrane Cofactor Protein
  • Membrane Glycoproteins
  • Protein Sorting Signals