Multiple system atrophy and progressive supranuclear palsy. Diminished striatal D2 dopamine receptor activity demonstrated by 123I-IBZM single photon emission computed tomography

Arch Neurol. 1993 May;50(5):513-6. doi: 10.1001/archneur.1993.00540050063017.

Abstract

Objective: To measure D2 dopamine receptors in the striatum in patients with multiple system atrophy and progressive supranuclear palsy by I 3-iodo-6-methoxybenzamide labeled with iodine I 123 (123I-IBZM) single photon emission computed tomography and differentiate them from control subjects.

Design: Survey with the following as retrospective criterion standards: (1) parkinsonism, (2) negative apomorphine test, and (3) no or only slight reaction to dopaminergic medication.

Setting: Ambulatory or hospitalized care in an academic referral center.

Patients and control subjects: Twenty-one patients with parkinsonism not responding to dopaminergic medication (17 with multiple system atrophy and four with progressive supranuclear palsy) and 21 control subjects without parkinsonism.

Intervention: In vivo imaging by single photon emission computed tomography using the D2 dopamine receptor specific radioligand 123I-IBZM.

Main outcome measure: Striatum/occipital cortex ratio of count rate density as semiquantitative measurement for striatal D2 dopamine receptor density.

Results: A highly significant loss of striatal uptake of 123I-IBZM was observed in the patients in comparison to the control subjects with little or no overlap between values.

Conclusions: The hypothesized loss of D2 receptors in multiple system atrophy has been confirmed. Use of 123I-IBZM single photon emission computed tomography may be a cost-effective alternative to positron emission tomography in the differential diagnosis of parkinsonism and in the selection of patients for dopaminergic therapy.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Atrophy
  • Benzamides* / pharmacokinetics
  • Central Nervous System / diagnostic imaging
  • Central Nervous System / metabolism
  • Central Nervous System / pathology*
  • Dopamine D2 Receptor Antagonists
  • Humans
  • Middle Aged
  • Parkinson Disease / diagnosis*
  • Parkinson Disease / diagnostic imaging
  • Parkinson Disease / metabolism
  • Pyrrolidines* / pharmacokinetics
  • Receptors, Dopamine D2 / metabolism*
  • Supranuclear Palsy, Progressive / diagnosis*
  • Supranuclear Palsy, Progressive / diagnostic imaging
  • Supranuclear Palsy, Progressive / metabolism
  • Tomography, Emission-Computed, Single-Photon*

Substances

  • Benzamides
  • Dopamine D2 Receptor Antagonists
  • Pyrrolidines
  • Receptors, Dopamine D2
  • 3-iodo-2-hydroxy-6-methoxy-N-((1-ethyl-2-pyrrolidinyl)methyl)benzamide