mdr 1 gene-expression and villin synthesis in a colon cancer cell line differentiated by sodium butyrate

Anticancer Res. 1993 Mar-Apr;13(2):487-90.

Abstract

Sodium butyrate (NaBu) but not dimethylsulfoxide (DMSO) induced the synthesis of villin, a protein of the brush border microvilli cytoskeleton, in a rat colon cancer cell line. Neither NaBu nor DMSO altered mdr 1-mRNA expression or multidrug resistance (MDR)--associated cellular transport of doxorubicin. These results show that mdr 1 gene expression and activity are independent of other brush border proteins induced by differentiating agents at the apical pole of the epithelial cell.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Biological Transport, Active / drug effects
  • Butyrates / pharmacology*
  • Butyric Acid
  • Carrier Proteins / biosynthesis*
  • Cell Differentiation / drug effects
  • Cell Differentiation / physiology
  • Cell Membrane / metabolism
  • Colonic Neoplasms / genetics*
  • Colonic Neoplasms / metabolism*
  • Colonic Neoplasms / pathology
  • Dimethyl Sulfoxide / pharmacology
  • Doxorubicin / pharmacokinetics
  • Drug Resistance / genetics*
  • Gene Expression / genetics*
  • Membrane Glycoproteins / metabolism
  • Membrane Glycoproteins / physiology
  • Microfilament Proteins / biosynthesis*
  • Rats
  • Rats, Inbred Strains
  • Tumor Cells, Cultured / drug effects

Substances

  • Butyrates
  • Carrier Proteins
  • Membrane Glycoproteins
  • Microfilament Proteins
  • villin
  • Butyric Acid
  • Doxorubicin
  • Dimethyl Sulfoxide