2,3-didehydro-2,4-dideoxy-4-guanidino-N-acetyl-D-neuraminic acid (4-guanidino-Neu5Ac2en) is a slow-binding inhibitor of sialidase from both influenza A virus and influenza B virus

Biochem Mol Biol Int. 1995 Jul;36(4):695-703.

Abstract

The effect of 2,3-didehydro-2,4-dideoxy-4-guanidino-N-acetyl-D-neuraminic acid (4-guanidino-Neu5Ac2en) on the sialidases from influenza virus reassortant X31 (which contains the sialidase from A/Aichi/2/68) and influenza virus B/Beijing/1/87 has been investigated. We find that 4-guanidino-Neu5Ac2en is a slow-binding inhibitor of both influenza A and influenza B virus sialidase, and that association and dissociation rate constants are almost identical for both enzymes. Furthermore, values for these rate constants are independent of whether purified enzyme or detergent-treated virus is used in the assays.

Publication types

  • Comparative Study

MeSH terms

  • Dose-Response Relationship, Drug
  • Enzyme Inhibitors / metabolism
  • Enzyme Inhibitors / pharmacology*
  • Guanidines
  • Humans
  • Influenza A virus / enzymology*
  • Influenza B virus / enzymology*
  • Kinetics
  • Neuraminidase / antagonists & inhibitors*
  • Neuraminidase / isolation & purification
  • Neuraminidase / metabolism
  • Pyrans
  • Sialic Acids / metabolism
  • Sialic Acids / pharmacology*
  • Species Specificity
  • Zanamivir

Substances

  • Enzyme Inhibitors
  • Guanidines
  • Pyrans
  • Sialic Acids
  • Neuraminidase
  • Zanamivir