Efficacy of two oral dose regimens of granisetron

Anticancer Res. 1995 Sep-Oct;15(5B):2287-90.

Abstract

Background: Most chemotherapic treatments are carried out on an outpatient basis. In such patients the prevention and control of emesis is important. Granisetron is a specific and extremely potent 5-HT3 antagonist available as an oral formulation. We have carried out an open randomized crossover study in patients receiving moderately emetogenic chemotherapy.

Materials and methods: 30 patients were randomized to receive one of the two oral dose regimens of GRAN. Treatment A = 1 mg of GRAN initially and 12 hours after the first; treatment B = a single 2 mg dose of GRAN. RESULTS. An overall good response for vomiting was reached in 70% and 86.7% respectively of patients receiving treatments A and B (p = 0.0625). Good response to nausea was reached in 73.3% of the patients with treatment A and in 76.7% with treatment B (p = 1). 68.3% of patients did not record chemoinduced emesis.

Conclusion: We believe that oral GRAN alone is an active and safe drug for the prevention of acute chemoinduced emesis.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial

MeSH terms

  • Administration, Oral
  • Adult
  • Aged
  • Antiemetics / administration & dosage*
  • Antineoplastic Agents / adverse effects*
  • Cross-Over Studies
  • Drug Administration Schedule
  • Female
  • Granisetron / administration & dosage*
  • Humans
  • Male
  • Middle Aged
  • Neoplasms / drug therapy*
  • Serotonin Antagonists / administration & dosage*
  • Vomiting / prevention & control*

Substances

  • Antiemetics
  • Antineoplastic Agents
  • Serotonin Antagonists
  • Granisetron