Amiloride inhibits meal-stimulated colonic absorption

J Surg Res. 1996 Feb 1;60(2):303-6. doi: 10.1006/jsre.1996.0047.

Abstract

Meal-stimulated colonic absorption has recently been described, but the cellular transport mechanisms mediating this response are unknown. The purpose of this study was to determine the contribution of Na+ transport pathways to colonic proabsorption. Distal colonic Thiry-Vella loops were constructed in six dogs. Absorption was measured by infusing the loops with a physiological electrolyte solution containing [14C] polyethylene glycol as the impermeant marker. In the first set of experiments, the dose dependence of amiloride-induced inhibition of basal colonic absorption was determined. In the second set of experiments the effect of amiloride, which inhibits both Na+ channels and Na+/H+ exchange in colonocytes, on meal-stimulated colonic absorption was determined. Luminal amiloride inhibited basal colonic absorption in a dose-dependent manner, with significant reductions in Na+ absorption occurring with concentrations of 10(-2)M and higher. Infusion with 10(-3)M amiloride, a concentration that did not alter basal absorption, resulted in significant reductions in postprandial water, Na+, and Cl- absorption. These results suggest that meal-stimulated colonic absorption is mediated, at last in part, by transcellular Na+ absorptive pathways.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amiloride / pharmacology*
  • Animals
  • Chlorides / metabolism
  • Colon / metabolism*
  • Dogs
  • Dose-Response Relationship, Drug
  • Female
  • Food
  • Intestinal Absorption / drug effects*
  • Sodium / metabolism
  • Sodium Channel Blockers*
  • Sodium-Hydrogen Exchangers / antagonists & inhibitors*

Substances

  • Chlorides
  • Sodium Channel Blockers
  • Sodium-Hydrogen Exchangers
  • Amiloride
  • Sodium