Inhibition of proliferation and clonal growth of human breast cancer cells by interleukin 13

Cancer Res. 1996 Aug 1;56(15):3583-8.

Abstract

We tested the influence of recombinant human interleukin (rhIL)-l3 and rhIL-4 on clonal growth of human breast cancer cell lines. rhIL-13 and rhIL-4 inhibited clonal growth of three of nine lines to approximately 50% of controls (ED50, 0.5 ng/ml). rhIl-13 reduced [3H]thymidine incorporation in all three cell lines: two showing a minor (84% and 83% of controls) and one showing a major response (25% of control). Both cytokines markedly reduced serum-induced G(0/1) exit (approximately 25% versus 60%). 125I-labeled interleukin (IL) 13 binding assays revealed high-affinity binding sites for IL-13 on two of the three responding cell lines (KD approximately 60 pM). (Y124D)IL-4 effectively antagonized all effects of rhIl-13 and rhIL-4, arguing for shared receptor components between them. However, neither rhIl-4 nor (Y124D) IL-4 could displace 125I-labeled IL-13 from binding, although unlabeled rhIL-13 effectively did so. Using reverse transcription-PCR, we studied the expression of the common gamma chain (gammac) in responding cell lines, putatively being shared between IL-4 receptor and IL-13 receptor; none of the three cell lines express gammac. In conclusion, we demonstrate antiproliferative effects of IL-4 and IL-13 on carcinoma cells which express IL-13 binding sites without participation of gammac.

MeSH terms

  • Animals
  • Antigens, CD / metabolism
  • Antineoplastic Agents / metabolism
  • Antineoplastic Agents / pharmacology*
  • Base Sequence
  • Binding Sites
  • Breast Neoplasms / drug therapy*
  • Breast Neoplasms / pathology*
  • CHO Cells
  • Cell Cycle / drug effects
  • Cell Division / drug effects
  • Cricetinae
  • DNA, Neoplasm / biosynthesis
  • Humans
  • Interleukin-13 / metabolism
  • Interleukin-13 / pharmacology*
  • Interleukin-13 Receptor alpha1 Subunit
  • Interleukin-4 / pharmacology
  • Iodine Radioisotopes
  • Molecular Sequence Data
  • Receptors, Interleukin / metabolism
  • Receptors, Interleukin-13
  • Receptors, Interleukin-4
  • Recombinant Proteins / pharmacology
  • Signal Transduction / drug effects
  • Signal Transduction / physiology
  • Tumor Cells, Cultured

Substances

  • Antigens, CD
  • Antineoplastic Agents
  • DNA, Neoplasm
  • IL13RA1 protein, human
  • Interleukin-13
  • Interleukin-13 Receptor alpha1 Subunit
  • Iodine Radioisotopes
  • Receptors, Interleukin
  • Receptors, Interleukin-13
  • Receptors, Interleukin-4
  • Recombinant Proteins
  • Interleukin-4