Itasetron (DAU 6215) prevents age-related memory deficits in the rat in a multiple choice avoidance task

Eur J Pharmacol. 1996 Sep 12;311(2-3):115-9. doi: 10.1016/0014-2999(96)00586-9.

Abstract

The effects of itasetron (endo-N-8-methyl-8-azabicyclo-[3.2.1.]-octo-3-yl) -2,3-dihydro-2-oxo-1 H-benzimidazole-1-carboxamide hydrochloride), a 5-HT3 receptor antagonist, on discrete memory abilities of the aged rat were assessed by using the multiple choice avoidance behavioral task. Chronic treatment with itasetron (i.p., 10 micrograms/kg, b.i.d., for three consecutive weeks), but not with vehicle, significantly improved retention abilities of the aged rats in this memory test. These results further support the important role of this 5-HT3 receptor antagonist in counteracting age-related memory degeneration in rodents.

MeSH terms

  • Age Factors
  • Aging / drug effects*
  • Aging / physiology
  • Animals
  • Avoidance Learning / drug effects*
  • Benzimidazoles / pharmacology*
  • Bridged Bicyclo Compounds, Heterocyclic / pharmacology*
  • Cognition / drug effects*
  • Male
  • Pain Measurement / drug effects
  • Psychomotor Performance / drug effects
  • Rats
  • Rats, Sprague-Dawley
  • Serotonin Antagonists / pharmacology*

Substances

  • Benzimidazoles
  • Bridged Bicyclo Compounds, Heterocyclic
  • Serotonin Antagonists
  • itasetron