Different collagenase gene products have different roles in degradation of type I collagen

J Biol Chem. 1996 Nov 8;271(45):28509-15. doi: 10.1074/jbc.271.45.28509.

Abstract

Vertebrate collagenases, matrix metalloproteinases (MMPs), cleave type I collagen at a single helical locus. We show here that rodent interstitial collagenases (MMP-13), but not human fibroblast collagenase (MMP-1), cleave type I collagen at an additional aminotelopeptide locus. Collagenase cDNAs and chimeric constructs in pET-3d, juxtaposing MMP-13 sequences amino-terminal to the active site in the catalytic domain and MMP-1 sequences carboxyl-terminal and vice versa, were expressed in Escherichia coli. Assays utilized collagen from wild type (+/+) mice or mice that carry a targeted mutation (r/r) that encodes substitutions in alpha1(I) chains that prevent collagenase cleavage at the helical locus. MMP-13 and chimeric molecules that contained the MMP-13 sequences amino-terminal to the active site cleaved (+/+) collagen at the helical locus and cleaved cross-linked (r/r) collagen in the aminotelopeptide (beta components converted to alpha chains). Human MMP-1 and chimeric MMP-1/MMP-13 with MMP-1 sequences amino-terminal to the active site cleaved collagen at the helical locus but not in the aminotelopeptide. All activities were inhibited by TIMP-1, 1,10-phenanthroline, and EDTA. Sequences in the distal two-thirds of the catalytic domain determine the aminotelopeptide-degrading capacity of MMP-13.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Collagen / metabolism*
  • Collagen Type I
  • Collagenases / genetics*
  • Collagenases / metabolism
  • Enzyme Inhibitors / pharmacology
  • Fibroblasts / enzymology
  • Glycoproteins / pharmacology
  • Humans
  • Matrix Metalloproteinase 1
  • Mice
  • Molecular Sequence Data
  • Mutagenesis, Site-Directed
  • Peptides / metabolism
  • Rats
  • Tissue Inhibitor of Metalloproteinases

Substances

  • Collagen Type I
  • Enzyme Inhibitors
  • Glycoproteins
  • Peptides
  • Tissue Inhibitor of Metalloproteinases
  • collagen type I trimeric cross-linked peptide
  • Collagen
  • Collagenases
  • Matrix Metalloproteinase 1