ts BCR-ABL kinase activation confers increased resistance to genotoxic damage via cell cycle block

Oncogene. 1996 Nov 21;13(10):2225-34.

Abstract

Using a temperature-sensitive mutant of the p210 BCR-ABL gene, transfected into a growth factor-dependent cell line (BaF3), we show that transient BCR-ABL kinase expression increases single cell and clonogenic resistance to apoptosis arising from genotoxic damage induced by ionizing radiation and VP-16/etoposide. This effect is achieved in the absence of any detectable changes in the levels of BCL-2, BAX or BCL-x proteins and is independent of proliferative, MAP kinase-dependent effects of BCR-ABL kinase. In contrast to parental cells that transiently arrest in G2 and then apoptose, p210 BaF3 cells show a pronounced and sustained G2 arrest following radiation coupled with enhanced phosphorylation of cdc2. A cell cycle block in early M phase induced by the mitotic spindle poison, nocodazole, does not provide protection from apoptosis. Reversal of G2 arrest by caffeine abolishes the protective effect of BCR-ABL kinase. These data provide further insight into the transforming properties of BCR-ABL and are relevant to the clinical intransigence of Ph-positive leukaemias.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents, Phytogenic / pharmacology
  • Apoptosis / drug effects*
  • Apoptosis / radiation effects
  • Caffeine / pharmacology
  • Cell Line / drug effects
  • Cell Line / radiation effects
  • Enzyme Induction / drug effects
  • Etoposide / pharmacology
  • Fusion Proteins, bcr-abl / metabolism*
  • G1 Phase / drug effects
  • G2 Phase / drug effects
  • G2 Phase / radiation effects
  • Interleukin-3 / pharmacology*
  • Mitosis / radiation effects
  • Phosphodiesterase Inhibitors / pharmacology
  • Phosphorylation
  • Protein Kinases / metabolism
  • Proto-Oncogene Proteins / metabolism
  • Proto-Oncogene Proteins c-bcl-2 / metabolism
  • Radiation Tolerance
  • Temperature
  • bcl-2-Associated X Protein
  • bcl-X Protein

Substances

  • Antineoplastic Agents, Phytogenic
  • Interleukin-3
  • Phosphodiesterase Inhibitors
  • Proto-Oncogene Proteins
  • Proto-Oncogene Proteins c-bcl-2
  • bcl-2-Associated X Protein
  • bcl-X Protein
  • Caffeine
  • Etoposide
  • Protein Kinases
  • Fusion Proteins, bcr-abl