Synthesis of aminothienopyrimidine and thienotriazolopyrimidine derivatives as potential anticonvulsant agents

Pharmazie. 1996 Jan;51(1):7-11.

Abstract

New aminothienopyrimidines and derivatives of the new thienotriazolopyrimidine ring system were synthesized to investigate their anticonvulsant activity. The tricyclic compounds 6a, c, e, f, m, o and p and two bicyclic derivatives 4f and 4o were tested. The pharmacological screening results are reported and discussed.

MeSH terms

  • Animals
  • Anticonvulsants / chemical synthesis*
  • Anticonvulsants / pharmacology
  • Chemical Phenomena
  • Chemistry, Physical
  • Male
  • Mice
  • Motor Activity / drug effects
  • Pyrimidines / chemical synthesis*
  • Pyrimidines / pharmacology
  • Rats
  • Seizures / prevention & control
  • Thiophenes / chemical synthesis*
  • Thiophenes / pharmacology
  • Triazoles / chemical synthesis*
  • Triazoles / pharmacology

Substances

  • Anticonvulsants
  • Pyrimidines
  • Thiophenes
  • Triazoles