Novel C-2 substituted carbapenem derivatives. Part I. Synthesis and biological activity of non-aromatic heterocyclic derivatives

J Antibiot (Tokyo). 1996 Dec;49(12):1258-65. doi: 10.7164/antibiotics.49.1258.

Abstract

A new series of carbapenems, having a saturated or partially unsaturated heterocycle at C-2, has been synthesised. The in vitro antibacterial activity of these compounds and their stability to human dehydropeptidase-1 (DHP-1) are described. The stereochemistry of the C-2 side-chain and the presence of a double bond in the heterocycle were shown to have significant effects on the stabilities of the compounds to DHP-1.

MeSH terms

  • Bacteria / drug effects*
  • Carbapenems / chemical synthesis*
  • Carbapenems / chemistry
  • Carbapenems / pharmacology*
  • Dipeptidases / metabolism
  • Humans
  • Microbial Sensitivity Tests
  • Molecular Conformation
  • Molecular Structure

Substances

  • Carbapenems
  • Dipeptidases
  • dipeptidase