HIV-1 entry and macrophage inflammatory protein-1beta-mediated signaling are independent functions of the chemokine receptor CCR5

J Biol Chem. 1997 Mar 14;272(11):6854-7. doi: 10.1074/jbc.272.11.6854.

Abstract

The human immunodeficiency virus type 1 (HIV-1) requires the presence of specific chemokine receptors in addition to CD4 to enter its target cell. The chemokine receptor CCR5 is used by macrophage-tropic strains of HIV-1, which predominate during the asymptomatic stages of infection. Here we investigate whether the ability of CCR5 to signal in response to its beta-chemokine ligands is necessary or sufficient for viral entry. Three CCR5 mutants with little or no ability to mobilize calcium in response to macrophage inflammatory protein-1beta could nonetheless support HIV-1 entry and the early steps in the virus life cycle with efficiencies comparable with those of wild-type CCR5. Conversely, a chimeric receptor with the N terminus of CCR2 replacing that of CCR5 responded to macrophage inflammatory protein-1beta and MCP-1 but did not efficiently support viral entry. These results demonstrate that chemokine signaling and HIV-1 entry are separable functions of CCR5 and that only viral entry requires the N-terminal domain of CCR5.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Cell Line
  • Chemokine CCL4
  • Dogs
  • HIV-1 / physiology*
  • Humans
  • Macrophage Inflammatory Proteins / metabolism*
  • Macrophages / metabolism*
  • Macrophages / virology
  • Mutation
  • Receptors, CCR5
  • Receptors, Cytokine / genetics
  • Receptors, Cytokine / metabolism*
  • Receptors, HIV / genetics
  • Receptors, HIV / metabolism*
  • Signal Transduction*
  • Virus Replication*

Substances

  • Chemokine CCL4
  • Macrophage Inflammatory Proteins
  • Receptors, CCR5
  • Receptors, Cytokine
  • Receptors, HIV