Effect of low dose oxandrolone and testosterone treatment on the pituitary-testicular and GH axes in boys with constitutional delay of growth and puberty

Clin Endocrinol (Oxf). 1997 Feb;46(2):209-16. doi: 10.1046/j.1365-2265.1997.t01-1-1150928.x.

Abstract

Objective: To investigate the effect of low dose oxandrolone and testosterone on the pituitary-testicular and GH-IGF-I axes.

Design: Prospective double-blind placebo-controlled trial.

Patients: Sixteen boys with constitutional delay of growth and puberty (CDGP) with testicular volumes 4-6 ml were randomized to 3 months treatment: Group 1 (n = 5), daily placebo: Group 2 (n = 5), 2.5 mg oxandrolone daily or Group 3 (n = 6), 50 mg testosterone monthly intramuscular injections with assessment (growth, pubertal development and overnight hormone profiles) at 0, 3, 6 and 12 months.

Main outcome measures: LH and GH profiles (15-minute samples) were analysed by peak detection (Pulsar), Fourier transformation and autocorrelation. Testosterone levels were measured hourly and insulin, SHBG, IGF-I, and IGFBP-3 levels at 0800 h. Statistical analysis was by multivariate analysis of variance for repeated measures.

Results: LH and testosterone parameters increased significantly with time in all 16 (LH AUC, P < 0.001; peak amplitude, P = 0.02; number of peaks, P = 0.02; testosterone AUC, P = 0.02; morning testosterone, P = 0.002). In Group 2, however, LH and testosterone parameters decreased at 3 months followed by a rebound increase at 6 and 12 months. SHBG levels were markedly reduced at 3 months (P = 0.006) and a wider range of dominant GH frequencies was present although GH AUC was not increased until 6 months, with an increase in GH pulse frequency but not amplitude. IGF-I levels were increased at both 3 and 12 months. In Group 3, pituitary-testicular suppression was not apparent, but GH levels increased with an increase in GH amplitude at 3 and 12 months.

Conclusion: Oxandrolone transiently suppressed the pituitary-testicular axis and altered GH pulsatility. Testosterone increased GH via amplitude modulation.

Publication types

  • Clinical Trial
  • Comparative Study
  • Randomized Controlled Trial

MeSH terms

  • Adolescent
  • Anabolic Agents / administration & dosage*
  • Anabolic Agents / therapeutic use
  • Double-Blind Method
  • Drug Administration Schedule
  • Growth Disorders / drug therapy*
  • Growth Hormone / metabolism
  • Humans
  • Luteinizing Hormone / metabolism
  • Male
  • Oxandrolone / administration & dosage*
  • Oxandrolone / therapeutic use
  • Pituitary Gland / drug effects
  • Pituitary Gland / metabolism
  • Prospective Studies
  • Puberty, Delayed / drug therapy*
  • Secretory Rate / drug effects
  • Testis / drug effects
  • Testis / metabolism
  • Testosterone / therapeutic use*

Substances

  • Anabolic Agents
  • Testosterone
  • Oxandrolone
  • Luteinizing Hormone
  • Growth Hormone